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GHSR

GHS-R,即生长激素促释放激素受体,别名Growth hormone secretagogue receptor type 1、GHS-R、GH-releasing peptide receptor。它是一种G蛋白偶联受体,主要在大脑、胃肠道和胰腺等组织中表达。GHS-R的作用机制是通过与生长激素促释放激素(GHRH)结合,激活Gαs蛋白,进而促进腺苷酸环化酶(AC)的活性,导致cAMP水平上升,激活蛋白激酶A(PKA),最终促进生长激素(GH)的释放。它不仅参与调节生长激素的分泌,影响生长发育,还与能量代谢、食欲控制、应激反应等多种生理过程有关。此外,GHS-R的活性也与某些疾病相关,例如肥胖和生长激素缺乏症。因此,GHS-R是内分泌学和代谢疾病研究中的一个重要靶点,针对GHS-R的药物开发有助于治疗相关疾病。

热销产品

GHSR Antibody (CSB-PA450853)

验证数据

CSB-PA450853

Western blot analysis of 1) Rat LiverTissue, 2)Jurkat with Ghrelin Receptor Rabbit pAb diluted at 1:2,000.

CSB-PA450853

Immunohistochemical analysis of paraffin-embedded Human BrainTissue using Ghrelin Receptor Rabbit pAb diluted at 1:200.

CSB-PA450853

Immunohistochemical analysis of paraffin-embedded Human Skin Tissue using Ghrelin Receptor Rabbit pAb diluted at 1:200.

GHSR Antibodies

GHSR for Homo sapiens (Human)

GHSR Proteins

GHSR Proteins for Oryctolagus cuniculus (Rabbit)

GHSR Proteins for Mustela putorius furo (European domestic ferret) (Mustela furo)

GHSR Proteins for Rattus norvegicus (Rat)

GHSR Proteins for Homo sapiens (Human)

GHSR Proteins for Sus scrofa (Pig)

GHSR Proteins for Mus musculus (Mouse)